Structure and stability of hexadentate complexes of ligands based on AAZTA for efficient PET labelling with gallium-68.

نویسندگان

  • Bradley P Waldron
  • David Parker
  • Carsten Burchardt
  • Dmitry S Yufit
  • Melanie Zimny
  • Frank Roesch
چکیده

Pre-organised tricarboxylate ligands based on 6-amino-perhydro-1,4-diazepine bind (68)Ga rapidly and selectively in acetate buffer at pH 4 to 7, forming kinetically stable complexes suitable for use in PET imaging.

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عنوان ژورنال:
  • Chemical communications

دوره 49 6  شماره 

صفحات  -

تاریخ انتشار 2013